Medicinal Chemistry (2003)

1. Arnusch, C.J. and Pieters, R.J. (2003). Solid phase synthesis of Vancomycine mimics European Journal of Organic Chemistry, 3131-3138.

2. Autar, R., Khan, A.S., Schad, M., Hacker, J., Liskamp, R.M.J and Pieters, R.J. (2003). Adhesion inhibition of F1C-fimbriated Escherichia coli and Pseudomonas aeruginosa PAK and PAO by multivalent carbohydrate ligands ChemBioChem 4, 1317-1325.

3. van Ameijde, J. and Liskamp, R.M. J. (2003). Synthesis of novel trivalent amino acid glycoconjugates based on the cyclotriveratrylene ( CTV') scaffold Organic & Biomolecular Chemistry 1, 2661-2669.

4. ♥ Catalina, M.I., Dekker, F.J., Liskamp, R.M.J., Versluis, C., Maier, C.S. and Heck, A.J.R. (2003). Structural analysis of high affinity divalent phosphopeptide hybrids of spleen tyrosine kinase International Journal of Mass Spectrometry and Ion Processes 228, 879-890.

5. Chamorro Pérez, M.C., & Liskamp, R.M.J. (2003). Approaches to the solid phase of a cyclotriveratrylene scaffold-based tripodal library as potential artificial receptors Journal of Combinatorial Chemistry 5, 794-801.

6. Dekker, F.J., Mol, N.J. de, Fischer, M.J.E. and Liskamp, R.M.J. (2003). Amino propynyl benzoic acid building block in rigid spacers of divalent ligands binding to the Syk SH2 domains with equally high affinity as the natural ligand Bioorganic & Medicinal Chemistry Letters 13, 1241-1244.

7. Dekker, F.J., Mol, N.J. de, Fischer, M.J.E., Kemmink, J. and Liskamp, R.M.J. (2003). Cyclic phosphopeptides for interference with Grb2 SH2 domain signal transduction prepared by ring-closing metathesis and phosphorylation Organic & Biomolecular Chemistry 1, 3297-3303.

8. Dekker, F.J., Mol, N.J. de, Bultinck, P.R.E., Kemmink, J., Hilbers, H.W. and Liskamp, R.M.J. (2003). Role of solution conformation and flexibility of short peptide ligands that bind to the p56lck SH2 domain Bioorganic & Medicinal Chemistry 11, 941-949.

9. Haan, E.C. de, Wauben, M.H.M., Wagenaar-Hilbers, J.P.A., Grosfeld-Stulemeyer, M.C., Rijkers, D.T.S., Moret, E.E. and Liskamp, R.M.J. (2003). Stabilization of peptide guinea pig myelin basic protein 72-85 by N-terminal acetylation - implications for immunological studies Molecular Immunology 40, 943-948.

10. ♥ Kol, M.A., Laak, A.N.C. van, Rijkers, D.T.S., Killian, J.A., Kroon, A.I.P.M. de and Kruijff, B. de (2003). Phospholipid flop induced by transmembrane peptides in model membranes is modulated by lipid composition Biochemistry 42, 231-237.

11. ♥ Kopitz, J., André, S., Reitzenstein, C. Von, Versluis, C., Kaltner, H., Pieters, R.J., Wasano, K., Kuwabara, I., Liu, F-T., Cantz, M., Heck, A.J.R. and Gabius, H-J. (2003). Homodimeric galectin-7 (p53-induced gene 1) is a negative growth regulator for human neuroblastoma cells Oncogene 22, 6277-6288.

12. Merkx, R.; Rijkers, D. T. S.; Kemmink, J. and Liskamp, R. M. J. (2003) Chemoselective coupling of peptide fragments using the Staudinger ligation. Tetrahedron Letters 44, 4515-4518.

13. de Mol, N.J. and Fischer, M.J.E. (2003) Applications of surface plasmon resonance (SPR) in ligand - receptor binding studies: affinity, kinetics and thermodynamics, Recent. Res. Devel. Anal. Biochem. 3, 1-19

14. Nijenhuis, W.A.J., Kruijtzer, J.A.W., Wanders, N., Vrinten, D.H., Garner, K.M., Schaaper, W.M.M., Meloen, R.H., Gispen, W.H., Liskamp, R.M.J. and Adan, R.A.H. (2003). Discovery and in vivo evaluation of new melanocortin-4 receptor-selective peptides Peptides 24, 271-280.

15. Vrasidas, I., Andre, S., Valentini, P., Bock, C., Lensch, M., Kaltner, H., Liskamp, R.M.J., Gabius, H-J., and Pieters, R.J. (2003). Rigidified multivalent lactose molecules and their interactions with mammalian galectins: a route to selective inhibitors Organic & Biomolecular Chemistry 1, 803-810.